Rifampin (rifampicin) vs Temsirolimus

Interacting Drugs
Rifampin (rifampicin)
vs
Temsirolimus
Security Level
Moderate, Consider therapy modification
Mechanism
Temsirolimus: Rifamycin Derivatives may decrease the serum concentration of Temsirolimus. Rifamycins will likely cause an even greater decrease in the concentration of the active metabolite sirolimus.
Management
Temsirolimus prescribing information recommends against coadministration with strong CYP3A4 inducers such as rifampin; however, if concurrent therapy is necessary, an increase in temsirolimus adult dose to 50 mg/week should be considered.

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Other Interactions of Rifampin (rifampicin)

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Other Interactions of Temsirolimus

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